Heterocyclic compounds

Inhibition of CXCL12/CXCR4 autocrine/paracrine loop reduces viability of human glioblastoma stem-like cells affecting self-renewal activity

Molecular Biology / Toxicology / Cancer stem cells / Humans / Glioblastoma / Animals / Akt / Cell Proliferation / Cell Survival / CM / Heterocyclic compounds / Down-Regulation / Animals / Akt / Cell Proliferation / Cell Survival / CM / Heterocyclic compounds / Down-Regulation

Asymmetric organocatalytic Michael addition of azlactones to cis-1,2-bis(phenylsulfonyl)ethene. A simple entry to quaternary alpha-amino acids

Organic Chemistry / Catalysis / Synthesis / New / Thiourea / CHEMICAL SCIENCES / Cyclization / Amino Acid Profile / Heterocyclic compounds / Organic Chemicals / CHEMICAL SCIENCES / Cyclization / Amino Acid Profile / Heterocyclic compounds / Organic Chemicals

Iridium N-Heterocyclic Carbene Complexes as Efficient Catalysts for Magnetization Transfer from para -Hydrogen

Hydrogen / Catalysis / Magnetic Resonance Spectroscopy / The / CHEMICAL SCIENCES / Iridium / Magnetics / Heterocyclic compounds / Iridium / Magnetics / Heterocyclic compounds

Inhibition of human immunodeficiency virus replication by a dual CCR5/CXCR4 antagonist

Virology / Calcium / HIV / Biological Sciences / Humans / Monoclonal Antibodies / Chemotaxis / Human immunodeficiency virus / Pyridines / Monoclonal Antibody / Antiviral Activity / Cell Surface Markers / Heterocyclic compounds / Low molecular weight / Monoclonal Antibodies / Chemotaxis / Human immunodeficiency virus / Pyridines / Monoclonal Antibody / Antiviral Activity / Cell Surface Markers / Heterocyclic compounds / Low molecular weight

Electronic Properties of 3, 3′‐Dimethyl‐5, 5′‐bis (1, 2, 4‐triazine): Towards Design of Supramolecular Arrangements of N‐Heterocyclic CuI Complexes

Algorithms / Chemistry / Quantum Theory / Copper / Temperature / Electronic properties / CHEMICAL SCIENCES / Electrons / X ray diffraction / Triazines / Organometallic Compounds / Ligands / Heterocyclic compounds / Static Electricity / Electronic properties / CHEMICAL SCIENCES / Electrons / X ray diffraction / Triazines / Organometallic Compounds / Ligands / Heterocyclic compounds / Static Electricity

Comparison of plasma and peritoneal concentrations of various categories of MRI blood pool agents in a murine experimental pharmacokinetic model

Magnetic Resonance Imaging / Multidisciplinary / Diffusion / Mice / Animals / Male / Gadolinium / Organometallic Compounds / Heterocyclic compounds / Contrast Media / Experimental Model / Male / Gadolinium / Organometallic Compounds / Heterocyclic compounds / Contrast Media / Experimental Model

Cyclic sulfamide γ-secretase inhibitors

Organic Chemistry / Mice / Animals / Protease Inhibitors / Structure activity Relationship / Brain Chemistry / Heterocyclic compounds / Brain Chemistry / Heterocyclic compounds

Preliminary ecotoxicological characterization of a new energetic substance, CL-20

Polymorphism / Ecotoxicology / Seed germination / Multidisciplinary / Toxicity / Nitrification / Oxidoreductases / Bacteria / Statistical Significance / Bioluminescence / Nitrogen / Luminescence / Marine Bacteria / Soil Microbiology / Environmental Impact / Vibrio / Analysis of Variance / Gramineae / Water soluble polymers / Toxicity Tests / Triazines / Acute Toxicity / Chlorophyta / Heterocyclic compounds / Toxicity Test / Soil Pollutants / Microbial community / Thallophyta / Nitrification / Oxidoreductases / Bacteria / Statistical Significance / Bioluminescence / Nitrogen / Luminescence / Marine Bacteria / Soil Microbiology / Environmental Impact / Vibrio / Analysis of Variance / Gramineae / Water soluble polymers / Toxicity Tests / Triazines / Acute Toxicity / Chlorophyta / Heterocyclic compounds / Toxicity Test / Soil Pollutants / Microbial community / Thallophyta

Novel heterocyclic glucocorticoids: in vitro profile and in vivo efficacy

Organic Chemistry / Cell line / Humans / Mice / Animals / Anti-inflammatory agents / Lipopolysaccharides / Rats / Tumor necrosis factor-alpha / Bioorganic and medicinal Chemistry / Heterocyclic compounds / Glucocorticoids / Anti-inflammatory agents / Lipopolysaccharides / Rats / Tumor necrosis factor-alpha / Bioorganic and medicinal Chemistry / Heterocyclic compounds / Glucocorticoids

Novel heterocyclic glucocorticoids: in vitro profile and in vivo efficacy

Organic Chemistry / Cell line / Humans / Mice / Animals / Anti-inflammatory agents / Lipopolysaccharides / Rats / Tumor necrosis factor-alpha / Bioorganic and medicinal Chemistry / Heterocyclic compounds / Glucocorticoids / Anti-inflammatory agents / Lipopolysaccharides / Rats / Tumor necrosis factor-alpha / Bioorganic and medicinal Chemistry / Heterocyclic compounds / Glucocorticoids

Novel heterocyclic glucocorticoids: in vitro profile and in vivo efficacy

Organic Chemistry / Cell line / Humans / Mice / Animals / Anti-inflammatory agents / Lipopolysaccharides / Rats / Tumor necrosis factor-alpha / Bioorganic and medicinal Chemistry / Heterocyclic compounds / Glucocorticoids / Anti-inflammatory agents / Lipopolysaccharides / Rats / Tumor necrosis factor-alpha / Bioorganic and medicinal Chemistry / Heterocyclic compounds / Glucocorticoids

Inhibition of CXCL12/CXCR4 autocrine/paracrine loop reduces viability of human glioblastoma stem-like cells affecting self-renewal activity

Molecular Biology / Toxicology / Cancer stem cells / Humans / Glioblastoma / Animals / Akt / Cell Proliferation / Cell Survival / CM / Heterocyclic compounds / Down-Regulation / Animals / Akt / Cell Proliferation / Cell Survival / CM / Heterocyclic compounds / Down-Regulation

Novel heterocyclic glucocorticoids: in vitro profile and in vivo efficacy

Organic Chemistry / Dissociation / Cell line / In Vitro / Humans / Mice / Alcohol / Animals / Anti-inflammatory agents / In Vivo / Lipopolysaccharides / Rats / Tumor necrosis factor-alpha / Bioorganic and medicinal Chemistry / Biological activity / Ligand / Heterocyclic compounds / Glucocorticoids / Mice / Alcohol / Animals / Anti-inflammatory agents / In Vivo / Lipopolysaccharides / Rats / Tumor necrosis factor-alpha / Bioorganic and medicinal Chemistry / Biological activity / Ligand / Heterocyclic compounds / Glucocorticoids

Novel polyazaheterocyclic systems: Synthesis, antitumor, and antimicrobial activities

Fungi / Cell line / Humans / Amines / Female / Antimicrobial activity / Bacteria / Anti-Bacterial Agents / HeLa cells / Antifungal Agents / Microbial Sensitivity Tests / Antitumor Activity / Antineoplastic Agents / Hydroxylamine / Heterocyclic compounds / Molecular Structure / Antimicrobial activity / Bacteria / Anti-Bacterial Agents / HeLa cells / Antifungal Agents / Microbial Sensitivity Tests / Antitumor Activity / Antineoplastic Agents / Hydroxylamine / Heterocyclic compounds / Molecular Structure

Preliminary ecotoxicological characterization of a new energetic substance, CL-20

Polymorphism / Ecotoxicology / Seed germination / Multidisciplinary / Toxicity / Nitrification / Oxidoreductases / Bacteria / Statistical Significance / Bioluminescence / Nitrogen / Luminescence / Green Algae / Marine Bacteria / Soil Microbiology / Environmental Impact / Vibrio / Analysis of Variance / Gramineae / Water soluble polymers / Toxicity Tests / Growth Inhibition / Triazines / Soil Microorganism / Vibrio Fischeri / Acute Toxicity / Chlorophyta / Lolium Perenne L. / Heterocyclic compounds / Toxicity Test / Soil Pollutants / Microbial community / Thallophyta / Medicago sativa / Adverse effect / Nitrification / Oxidoreductases / Bacteria / Statistical Significance / Bioluminescence / Nitrogen / Luminescence / Green Algae / Marine Bacteria / Soil Microbiology / Environmental Impact / Vibrio / Analysis of Variance / Gramineae / Water soluble polymers / Toxicity Tests / Growth Inhibition / Triazines / Soil Microorganism / Vibrio Fischeri / Acute Toxicity / Chlorophyta / Lolium Perenne L. / Heterocyclic compounds / Toxicity Test / Soil Pollutants / Microbial community / Thallophyta / Medicago sativa / Adverse effect
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